CP-809101 hydrochloride

Short Summary : 5-HT2C receptor agonist, potent and selective

Category : Neuroscience|5-HT Receptor

Purity : 0.98

CAS Number : 1215721-40-6

Formula : C15H18Cl2N4O

Molecular Weight : 341.24

SMILE : C1CN(CCN1)C2=CN=CC(=N2)OCC3=CC(=CC=C3)Cl.Cl

Solubility : Soluble in DMSO > 10 mM

Storage : Store at -20°C

Description : CP-809101 is a potent and selective 5-HT2C receptor agonist (pEC50 values are 9.96, 7.19 and 6.81 for human 5-HT2C, 5-HT2B and 5-HT2A receptors respectively). CP-809101 displays antipsychotic activity; suppresses condition avoidance responding (CAR) and inhibits PCP and amphetamine-stimulated hyperactivity in rats following subcutaneous administration.

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