GDC-0980

GDC-0980 (Apitolisib, GNE 390, RG 7422) is a potent, selective, orally available class I PI3K/mTOR inhibitor with IC50 of 5 nM/27 nM/7 nM/14 nM for PI3K?/?/?/?, inhibits mTOR inhibitor with Ki of 17 nM.

Target : PI3K

CAS Number : 1032754-93-0

Formula Weight : 498.6011

Molecular Formula : C23H30N8O3S

Purity : >98% (HPLC)

Storage : (-20?)

Shipping Conditions : With Ice Pack

Stability : ? 2 years

Research use only, not for human use.