Avapritinib

Avapritinib (BLU-285) is a potent and highly selective inhibitor of mutant KIT and PDGFR? with IC50 of 0.6, 0.27 and 0.24 nM for KIT del557-558, KIT D816V and PDGFRA D842V, respectively.

Target : c-Kit

CAS Number : 1703793-34-3

Formula Weight : 498.57

Molecular Formula : C26H27FN10

Purity : >98% (HPLC)

Storage : (-20?)

Shipping Conditions : With Ice Pack

Stability : ? 2 years

Research use only, not for human use.