RVX-208

RVX-208 is a potent BET bromodomain inhibitor with IC50 of 0.510 ?M for BD2 in a cell-free assay, about 170-fold selectivity over BD1. Phase 2.

Target : Epigenetic Reader Domain

CAS Number : 1044870-39-4

Formula Weight : 370.4

Molecular Formula : C20H22N2O5

Purity : >98%(HPLC)

Storage : (-20?)

Shipping Conditions : With Ice Pack

Stability : ? 2 years

Research use only, not for human use.